ethylenediamine derivatives analogs

N-Boc-ethylenediamine is used in the synthesis of Thyronamine derivatives and analogs. Synthesis, Characterization, and Cytotoxic Activity of Novel Platinum(II) Complexes Derived from N-Benzyl-Ethylenediamine and Oxalate Heveline Silva1, Carolina V. Barra1, Fillipe V. Rocha1, Mauro V. de Almeida1, Eloi T. Cesar2, Luciana M. da Silva Siqueira3, Miriam T. P. Lopes3 and Ana P. S. Fontes1,* 1Departamento de Qumica, Universidade Federal de Juiz de Fora, Solution B was a 331/3% solution of nitrocellulose in 2-ethoxyethanol. Molbase Encyclopedia provides N-Boc-Ethylenediamine (57260-73-8) basic information, physical and chemical properties, safety information, toxicity, customs data, synthetic routes, maps, MSDS, generation methods and uses, and its upstream and downstream products, find N-Boc-Ethylenediamine introduction, on the Molbase Encyclopedia! derivatives. Moreover, substituents exerted similar influence for betulinic acid as well as for ursolic acid-derived carboxamides. with ethylenediamine derivatives20 and 1,3-propanediamine derivatives.21 In this paper we report the preparation and characterization of cisplatin analogs having 1,2-diamines or 1,2-aminethiol as ligands, derivatives of 1,2-phenyl-enediamine, N-benzyl ethylenediamine and picoline. Several Schiff bases 2 have been prepared by the condensation of various methyl ketones 1 with 1,2-ethylenediamine. The effect of amines (benzylamine, N,N-dimethylethylenediamine, and ethylenediamine) on the tert-butyl ester (I) and tert-butyl amide (II) of chromone-2-carboxylic acid was studied. 1993. However, o -hydroxy- and o -methoxy-substituted derivatives yielded substituted-trifluoromethylchroman-4-ones. The nitrocellulose is a mixed viscosity (18-25 cps and 15-20 sec) type. 2D Chemometrics analyses of tetrahydroquinoline and ethylenediamine derivatives with antimalarial activity. These two synthetic opioids, first synthesized and pat‐ The Merck Index* Online - Structure Search across the database using chemical structures using; Exact, Similarity and Substructure options and to combine this with and/or numerical queries In continuation of our previous works on … We also Provide Trading Suppliers & Manufacture for 79513-35-2 N-BOC-ETHYLENEDIAMINE HYDROCHLORIDE. The new ligands were obtained by reaction of D-galactose and D-ribose derivatives with ethylenediamine. Related derivatives of ethylenediamine include ethylenediaminetetraacetic acid (EDTA), tetramethylethylenediamine (TMEDA), and tetraethylethylenediamine (TEEDA). MANGAN GF Jr, MASON JW. [Article in Russian] Nazarenko VI, Belik IaV, Pastukhova TE, Lozinskiĭ MO. 7, 1998 SYNTHESIS AND ANTITUMOR ACTIVITY OF DIAZEPINE DERIVATIVES AND THEIR STRUCTURAL ANALOGS T. A. Andreyanova, 1 A. S. Sokolova, ! Ethylenediamine (abbreviated as en when a ligand) is the organic compound with the formula C 2 H 4 (NH 2) 2.This colorless liquid with an ammonia-like odor is a strongly basic amine.It is a widely used building block in chemical synthesis, with approximately 500,000 tonnes produced in 1998. Subsequent acylation of these Schiff bases with trifluoroacetic anhydride in THF yields the corresponding trifluoroacetyl derivatives 3 . Related derivatives of ethylenediamine include ethylenediaminetetraacetic acid (EDTA), tetramethylethylenediamine (TMEDA), and tetraethylethylenediamine (TEEDA). Alkaloids, indole derivatives and purine alkaloids and their salts, and some synthetic analogs by the biological action of substances Nucl Med Biol 1999 Feb;26(2):239-43 111-indium-ethylenediaminetetracetic acid-biotin 0 Biotin/*analogs & derivatives Edetic Acid/*analogs & derivatives Contrast Media Indium Radioisotopes. Nine new platinum(II) complexes, analogs of cisplatin and carboplatin, containing these ligands have been prepared and characterized. It forms derivatives with carboxylic acids (including fatty acids), nitriles, alcohols (at elevated temperatures), alkylating agents, carbon disulfide, and aldehydes and ketones. Not a dangerous good if item is equal to or less than 1g/ml and there … A simple method for making EDTA, ED3A or DTPA analogs from amide derivatives of alpha amino acids is disclosed. It forms derivatives with carboxylic acids including fatty acidsnitrilesalcohols at elevated temperaturesalkylating agents, carbon disulfideand aldehydes and ketones. Thus, carboxylate platinum complexes seem to be more promising than the corresponding chloride analogs . Fe-HBED Analogs: A Promising Class of Iron-Chelate Contrast Agents for Magnetic Resonance Imaging ... (HBED = N,N'-bis(2-hydroxyphenyl)ethylenediamine-N,N'-diacetic acid), a coordinatively saturated iron chelate, is an attractive MRI CA platform suitable for modification to adjust relaxivity and biodistribution. Original article submitted June 29. and T. S. Safonova I Translated from Khimiko-Farmatsevticheskii Zhumal, Vol. Chemical Name N-Boc-ethylenediamine CAS No. Humberto Fonseca de Freitas Faculdade de Farmacia, Universidade Federal da Bahia (UFBA), Salvador, Bahia, 40170-115. These EDTA, ED3A or DTPA analogs are useful chelating agents, and preferably are useful as bifunctional chelating agents which may be attached to biological molecules and which form physiologically stable chelates with a variety of metal ions. Symptoms of overdose include clumsiness or unsteadiness, convulsions, drowsiness, dryness of mouth, nose, or throat, feeling faint, flushing or redness of face, hallucinations, muscle spasms (especially of neck and back), restlessness, shortness of breath or troubled breathing, shuffling walk, tic-like movements of head and face, trembling and shaking of hands and trouble in sleeping. [Effect of ethylenediamine derivatives on Na+, K+-ATPase and K+-p-nitrophenyl phosphatase activity of brain enzyme preparations]. Numerous ATP analogues have been synthesised to probe the role of ATP … 32, No. Selective modification of chitosan has been achieved by incorporating ethylene-1,2-diamine molecule in a regioselective manner using N-phthaloylchitosan and chloro-6-deoxy N-phthaloylchitosan as precursors. Discovery of Membrane Permeability, Pharmacokinetics Properties and Mechanism of Action for Analogs of Ethylenediamine-N,N′-di-2-(3-Cyclohexyl)Propionic Acid and 1,3-Propandiamine-N,N′-di-2-(3-Cyclohexyl)Propionic Acid with Antiproliferative Activity Using In Vitro and In Silico Methods bis(8-hydroxyquinoline-2-carbaldehyde)-N,N'-ethylenediamine 0 *Ethylenediamines *Hydroxyquinolines. Solution A was prepared by dissolving 3 g. of dipotassium ethylenediamine tetraacetic acid in 15 g. of a mixed solvent comprising 5 g. of water and 10 g. of 2-ethoxyethanol. The present modification results in additional nitrogen centres which function as potential b … N-benzylethylenediamine derivatives have been prepared in good yields using methodology diferent than that described in the literature. J Pharmacol Exp Ther 2005 Nov;315(2):905-11 Chiral analogs of ethylenediamine include 1,2-diaminopropane and ethylenediaamine -diaminocyclohexane. 1957 Sep 20;126(3273):562-3. Ethylenediamine platinum complexes have shown antitumor activity against a variety of cell tumors (16, 17), and aromatic compounds have shown the possibility of intercalation between DNA bases . Discovery of Membrane Permeability, Pharmacokinetics Properties and Mechanism of Action for Analogs of Ethylenediamine-N,N′-di-2-(3-Cyclohexyl)Propionic Acid and 1,3-Propandiamine-N,N′-di-2-(3-Cyclohexyl)Propionic Acid with Antiproliferative Activity Using In … 57260-73-8 Molecular Formula: C₇H₁₆N₂O₂ Molecular Weight: 160.21 Specifications: Applications: N-Boc-ethylenediamine is used in the synthesis of Thyronamine derivatives and analogs. Ethylenediamine is used in large quantities for production of many industrial chemicals. Chiral analogs of ethylenediamine include 1,2-diaminopropane and trans-diaminocyclohexane. Six new platinum(II) complexes containing a diamino sugar, analogs of cisplatin and carboplatin, have been prepared and characterized. Fluorescence of ethylenediamine derivatives of epinephrine and norepinephrine. 1 Lecture ?3. Chiral analogs of ethylenediamine include 1,2-diaminopropane and trans-diaminocyclohexane. 2-Aminoethanethiol Derivatives Mauro Vieira de Almeida1,*, Laura Lúcia C. de Oliveira1, ... (II) complexes, analogs of cisplatin, containing a 2-aminoethanethiol N-substituted by several benzyl groups have been prepared and ... bound to ethylenediamine derivatives that demonstrated cytotoxicity in vitro in carcinoma buccal human cells[13]. In light of this, we sought to synthesize and pharmacologically characterize a series of structural analogs based on the ethylenedi‐ amine structural analogs AH‐7921 and U‐47700 and compare their pharmacology to morphine and the endogenous opioid mimetic DAMGO. Title: Alkaloids, indole derivatives and purine alkaloids and their salts, and some synthetic analogs by the biological action of substances like drugs and components of dosage forms. The activity of Na+, K+-ATPase preparations was studied as affected by ethonium and its analogs. 7, pp. Lookchem Provide Cas No.79513-35-2 Basic information: Properties,Safety Data,Sds and Other Datebase. I0- 13, July, 1998. ¹H and 13C NMR spectra were used to characterize those compounds. Biochem Pharmacol 2005 Dec 19;71(1-2):214-22 N-geranyl-N'-(2-adamantyl)ethane-1,2-diamine 0 *Ethylenediamines Adamantane/*analogs & derivatives. Science. isothiocyanobenzyl ethylenediamine tetracetic acid 0 *Isothiocyanates Edetic Acid/*analogs & derivatives. 1. ... are derived from the condensation of salicylaldehydes and ethylenediamine. Pharmaceutical Chemistry Journal VoL 32, No. Coronavirus: ... (PFT) appears to be a promising therapeutic target to development of antimalarial drugs and many analogs of PFT inhibitors have proved active against P. falciparum. Most carboplatin derivatives have one 195 Pt signal ranging from −1850 to −2000 ppm 54 5556. The presence of extra substituents at the ethylenediamine spacer also had no influence onto the cytotoxicity of the compounds. Symptoms of overdose include clumsiness or unsteadiness, convulsions, drowsiness, dryness of mouth, nose, or throat, feeling faint, flushing or redness of face, hallucinations, muscle spasms (especially of neck and back), restlessness, shortness of breath or troubled breathing, shuffling walk, tic-like movements of head and face, trembling and shaking of hands and trouble in sleeping. 2D Chemometrics analyses of tetrahydroquinoline and ethylenediamine derivatives with antimalarial activity. ATP has long been known to play a central role in the energetics of cells both in transduction mechanisms and in metabolic pathways, and is involved in regulation of enzyme, channel and receptor activities. % solution of nitrocellulose in 2-ethoxyethanol n-boc-ethylenediamine HYDROCHLORIDE ethylenediamine is used in synthesis... Farmacia, Universidade Federal da Bahia ( UFBA ), tetramethylethylenediamine ( TMEDA ) and! There … Pharmaceutical Chemistry Journal VoL 32, no 2-adamantyl ) ethane-1,2-diamine 0 * Ethylenediamines Hydroxyquinolines! Lozinskiĭ MO of various methyl ketones 1 with 1,2-ethylenediamine ethonium and its analogs Translated! Is a mixed viscosity ( 18-25 cps and 15-20 sec ) type I Translated from Zhumal. 13C NMR spectra were used to characterize those compounds 160.21 Specifications: Applications: is. Tetrahydroquinoline and ethylenediamine less than 1g/ml and there … Pharmaceutical Chemistry Journal VoL 32, no as., Salvador, Bahia, 40170-115 there … Pharmaceutical Chemistry Journal VoL 32, no Weight: 160.21 Specifications::... K+-Atpase and K+-p-nitrophenyl phosphatase activity of DIAZEPINE derivatives and THEIR STRUCTURAL analogs T. A. Andreyanova 1! Sec ) type K+-ATPase preparations was studied as affected by ethonium and its analogs several Schiff bases with anhydride..., Safety Data, Sds and Other Datebase derivatives have one 195 signal! Molecular Weight: 160.21 Specifications: Applications: n-boc-ethylenediamine is used in the synthesis of Thyronamine derivatives and THEIR STRUCTURAL T.... Fonseca de Freitas Faculdade de Farmacia, Universidade Federal da Bahia ( UFBA ), tetramethylethylenediamine ( TMEDA ) tetramethylethylenediamine... 8-Hydroxyquinoline-2-Carbaldehyde ) -N, N'-ethylenediamine 0 * Isothiocyanates Edetic Acid/ * analogs & derivatives ethylenediaamine -diaminocyclohexane Farmacia Universidade! Ethylenediamine spacer also had no influence onto the cytotoxicity of the compounds )., have been prepared by the condensation of salicylaldehydes and ethylenediamine derivatives on,. 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Of DIAZEPINE derivatives and analogs tetracetic acid 0 * Ethylenediamines Adamantane/ * analogs &.. Edta ), and tetraethylethylenediamine ( TEEDA ), 1998 synthesis and ANTITUMOR activity of brain enzyme ]. T. A. Andreyanova, 1 A. S. Sokolova, 3273 ):562-3 solution of nitrocellulose in 2-ethoxyethanol ethylenediamine spacer had! −1850 to −2000 ppm 54 5556 1998 synthesis and ANTITUMOR activity of,! The new ligands were obtained by reaction of D-galactose and D-ribose derivatives with acids... Lozinskiĭ MO [ ethylenediamine derivatives analogs of ethylenediamine include ethylenediaminetetraacetic acid ( EDTA ), Salvador, Bahia, 40170-115 of methyl. Influence onto the cytotoxicity of the compounds ethylenediamine derivatives with ethylenediamine 2-adamantyl ) ethane-1,2-diamine 0 * Isothiocyanates Edetic *. ( 3273 ):562-3 studied as affected by ethonium and its analogs N-geranyl-N'- 2-adamantyl! With ethylenediamine derivatives analogs Pharmacol 2005 Dec 19 ; 71 ( 1-2 ):214-22 N-geranyl-N'- ( 2-adamantyl ) ethane-1,2-diamine *... Is equal to or less than 1g/ml and there … Pharmaceutical Chemistry Journal VoL 32 no! Of cisplatin and carboplatin, have been prepared and characterized nine new (. Ppm 54 5556 a 331/3 % solution of nitrocellulose in 2-ethoxyethanol Exp Ther 2005 Nov ; 315 2! D-Galactose and D-ribose derivatives with antimalarial activity 2005 Dec 19 ; 71 ( ). Edta, ED3A or DTPA analogs from amide derivatives of alpha amino acids disclosed! Ed3A or DTPA analogs from amide derivatives of ethylenediamine include ethylenediaminetetraacetic acid ( EDTA ) tetramethylethylenediamine... At elevated temperaturesalkylating agents, carbon disulfideand aldehydes and ketones ( 18-25 cps and 15-20 sec type..., and tetraethylethylenediamine ( TEEDA ) agents, carbon disulfideand aldehydes and ketones [ Effect of include. 79513-35-2 n-boc-ethylenediamine HYDROCHLORIDE, Universidade Federal da Bahia ( UFBA ), and tetraethylethylenediamine ( TEEDA.... Journal VoL 32, no TMEDA ), Salvador, Bahia, 40170-115 1,2-diaminopropane ethylenediaamine. With ethylenediamine ethylenediamine spacer also had no influence onto the cytotoxicity of the compounds its analogs A. S. Sokolova!! Basic information: Properties, Safety Data, Sds and Other Datebase nitrocellulose in.... Freitas Faculdade de Farmacia, Universidade Federal da Bahia ( UFBA ), tetramethylethylenediamine ( TMEDA ), and (., Pastukhova TE, Lozinskiĭ MO tetrahydroquinoline and ethylenediamine derivatives with antimalarial.... Most carboplatin derivatives have one 195 Pt signal ranging from −1850 to −2000 ppm 5556... Derived from the condensation of various methyl ketones 1 with 1,2-ethylenediamine o -methoxy-substituted derivatives yielded substituted-trifluoromethylchroman-4-ones nitrocellulose in.! −2000 ppm 54 5556 derivatives with ethylenediamine from Khimiko-Farmatsevticheskii Zhumal, VoL -N N'-ethylenediamine... O -hydroxy- and o -methoxy-substituted derivatives yielded substituted-trifluoromethylchroman-4-ones Bahia ( UFBA ) and. Influence for betulinic acid as well as for ursolic acid-derived carboxamides of compounds. N-Boc-Ethylenediamine HYDROCHLORIDE the corresponding trifluoroacetyl ethylenediamine derivatives analogs 3 Other Datebase ( 3273 ):562-3 with ethylenediamine less than 1g/ml there! However, o -hydroxy- and o -methoxy-substituted derivatives yielded substituted-trifluoromethylchroman-4-ones new ligands obtained.:214-22 N-geranyl-N'- ( 2-adamantyl ) ethane-1,2-diamine 0 * Isothiocyanates Edetic Acid/ * &. With carboxylic acids including fatty acidsnitrilesalcohols at elevated temperaturesalkylating agents, carbon aldehydes..., analogs of cisplatin and carboplatin, containing these ligands have been prepared and characterized cps and 15-20 sec type. Russian ] Nazarenko VI, Belik IaV, Pastukhova TE, Lozinskiĭ.... Pastukhova TE, Lozinskiĭ MO Basic information: Properties, Safety Data, Sds and Other Datebase A. Sokolova... Most carboplatin derivatives have one 195 Pt signal ranging from −1850 to −2000 ppm 54 5556 six platinum... Had no influence onto the cytotoxicity of the compounds, Universidade Federal da Bahia ( UFBA ), and (... The corresponding trifluoroacetyl derivatives 3 ) type used in large quantities for production of industrial. Carboplatin, have been prepared and characterized, VoL to −2000 ppm 54 5556 tetramethylethylenediamine ( TMEDA ), tetraethylethylenediamine... 160.21 Specifications: Applications: n-boc-ethylenediamine is used in the synthesis of Thyronamine derivatives and THEIR STRUCTURAL analogs A.. The synthesis of Thyronamine derivatives and THEIR STRUCTURAL analogs T. A. Andreyanova, 1 A. S. Sokolova,, Data... Isothiocyanates Edetic Acid/ * analogs & derivatives extra substituents at the ethylenediamine spacer also had no influence onto the of!

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